Abbas Shafiee, Iranian pharmaceutical and organic chemist (01 September 1937 – 15 June 2016)

Authored 473 papers, 8 essays and 5 books

CONTRIBUTIONS

With M. Madhavi, S. Dianat, B. Khavari, S. Moghini et al. Synthesis and biological evaluation of novel imidazo-pyrimidin-3-amines as anticancer agents. Chem. Biol. Drug Des. 89(5):797-805, 2017

With R. Hariri, Z. Ashfar, M. Madhavi, M. Safavi et al. Novel tacrine-based pyrano[3’,4’,5, 6]pyrano[2,3-b]quinolones:synthesis and cholinesterase inhibitory activity. Arch. Pharm. 349(12):915-24, 2016 

With S. Dianat, S. Moghimi, M. Madhavi, H. Nadri et al. Quinoline-based imidazole-fused heterocycles as new inhibitors of 15-lipoxygenase. J. Enzyme Inhib. Med. Chem. 31 (Sup3):205-9, 2016

With M. Alipour, M. Khoobi, A. Foroumadi, H. Nadri et al. Novel coumarin derivatives bearing N-benzyl pyridinium moiety: potent and dual binding site acetylcholinesterase inhibitors (2012)

With A. Zarghi, Z. Hajimahdi, S. Mohebbi, H. Rashidi, S. Mozaffari, S. Sarraf, M. Faizi & S.A. Tabatabaee. Design and synthesis of new 2-substituted-5-[2-(2-halobenzyloxy)phenyl]-1,3,4-oxadiazoles as anticonvulsant agents. Chem. Pharm. Bull. (2008)

With M. Amini & L. Navidpour. Synthesis and antitubercular activity of new N, N-diaryl-4-(4,5-dichloroimidazole-2-yl)-1,4-dihydro-2,6- dimethyl-3,5-pyridinedicarboxamides. DARU 16:9-12, 2008

With S. Rabajalian, A. Foroumadi & S. Emami. Functionalized N(2-oxyiminoethyl) piperazinyl quinolones as new cytotoxic agents. J. Pharm. Pharmac. Sci. (2007)

With E. Souri & H. Jalalizadeh. Optimization of an HPLC method for determination of gabapentin in dosage forms through derivatization with 1-fluoro-2,4-dinitrobenzene. Chem. Pharm. Bull. (2007)

With N. Hadj-Esfandiari, L. Navidpour, H. Shadnia, M. Amini, N. Samadi & M.A.Faramarzi. Synthesis, antibacterial activity, and quantitative structure-activity relationships of new (Z)-2-(nitroimidazolylmethylene)-3(2H)-benzofuranone derivatives. Bioorg Med Chem Lett (2007)

With L. Amini & L. Navidpour. Synthesis and antitubercular activity of new N,N-diaryl-4-(4,5-dichloroimidazole-2-yl)-1,4-dihydro-2,6-dimethyl-3,5-pyridinedicarboxamides. DARU 16 (2008)

With A. Foroumadi, N. Mohammadhosseini, S. Emami, B. Letafat, M.A. Faramarzi & N. Samadi. Synthesis and antibacterial activity of new 7-piperazinyl-quinolones containing a functionalized 2-(furan-3-yl)ethyl moiety. Archiv der Pharmazie (2007)

With B. Letafat, S. Emami, N. Mohammadhosseini, M.A. Faramarzi, N. Samadi & A. Foroumadi. Synthesis and antibacterial activity of new N-[2-(thiophen-3-yl)ethyl] piperazinyl quinolones. Chem. Pharm. Bull. (2007)

With N. Hadj- Esfandiari, L. Navidpour, H. Shadnia, M. Amini, N. Samadi & M. A. Faramarzi. Synthesis, antibacterial activity, and quantitative structure-activity relationships of new (Z)-2-(nitroimidazolylmethlene)-3(2H)-bezofuranone derivatives. Bioorg. Med Chem Lett 17:6354-6363, 2007

With A. Foroumadi, L. Firoozpour, N. Nematollahi & A. Asadipour. Synthesis of New Fluroquinolones Containing a N-[5-(Fluorobenzylthio)- 1,3,4-thiadiazol-2-yl]piperazine moiety. Asian J. Chem. 19(6); 4547-52, 2007

With K. M. Taghi-Ganji, Sh. Ghodsi, A. Alipour, M. Amini & M. Hosseini. Synthesis and Characterization of Some New 1,4-Dihydropyridine Derivatives Containing Dichlorothiazolyl Substituents. Asian J. Chem. 19(4):2521-6, 2007

With N. Daryabari, T. Akbarzadeh, M. Amini, R. Miri & H. Mirkhani. Synthesis and Calcium Channel Antagonist Activities of New Derivatives of Dialkyl 1,4-Dihydro-26-dimethyl-4-(5-phenylisoxazol-3-yl)pyridine, 3,5- dicarboxylates. J. Iran. Chem. Soc. 4(1):30-6, 2007

With S. Rejabalian, A. Foroumadi & S. Emami. Functionalized N-(2-oxyiminoethyl)piperzinyul quinolones as new cytotoxic agents. J. Pharm. Pharmaceut. Sci 10(2):123-128, 2007

With M.Z. Kassaee & A.R. Bekhradnia. Synthesis of novel 3,4 diaryl-1H-pyrroles. J. Heteroc. Chem. 44(2):471-4, 2007

With L. Navidpour, M. Amini & H. Shafaroodi. A Convenient Synthesis of 5-Alkylthio-3,4-diarylisoxazoles by Palladium- Catalyzed Coupling Reactions. J. Heterocyclic Chem 44:471, 2007

With L. Navidpour, M. Amini, H. Shafaroodi, K. Abdi, M.H. Ghahremani & A.R. Dehpour. Design and synthesis of new water-soluble tetrazolide derivatives of celecoxib and rofecoxib as selective cyclooxygenase-2 (COX-2) inhibitors. Bioorg. Med. Chem. Lett. (2006)

With S. Emami & A. Foroumadi. Structural features of new quinolones and relationship to antibacterial activity against Gram-positive bacteria. Mini reviews Med. Chem. (2006)

With A. Davvod, N. Mansouri, A. R. Dehpour, H. Shafaroudi & E. Alipour. Design, synthesis, and calcium channel antagonist activity of new 1,4-dihydropyridines containing 4-(5)-chloro-2-ethyl-5-(4)-imidazolyl substituent. Arch. Pharm. (2006)

With S. Emami, A. Kebriaeezadeh & M.J. Zamani. Azolychromans as a novel scaffold for anticonvulsant activity. Bioorg. Med. Chem. Lett. 16:1804-6, 2006

With S. Ghodsi, M. Amini, R. Miri, K.M. Tagi-Ganji, J. Hosseini & H. Mirkhani. The Synthesis and Characterization New Asymmetrical Dihydropyridine Derivatives Containing a 2,4-Dichloro-5-Thiazolyl Substituent. Phosphorus, Sulfur & Silicon. 181:2435-44, 2006

With S. R.A. Ali Khalaj, M. Daneshtalab, A. Madadkar-Sobhani, S. Fouladdel & E. Azizi. Anti-tumor Activity of New quinolone Derivatives in Human Breast Cancer T47D Cells. Int. J. Cancer Res. 2(2):102-8, 2006

With A. Zarghi, M. Faizi, B. Shafaghi, A. Ahadian, H.R. Khojastehpoor, V. Zanganeh & S.A. Tabatabai. Design and synthesis of new 2-substituted-5-(2-benzylthiophenyl)-1,3,4-oxadiazoles as benzodiazepine receptor agonists. Bioorg. Med. Chem. Lett. (2005)

With A. Zarghi, S.A. Tabatabai, M. Faizi, A. Ahadian, P. Navabi & V. Zanganeh. Synthesis and anticonvulsant activity of new 2-substituted-5-(2-benzyloxyphenyl)-1,3,4-oxadiazoles. Bioorg. Med. Chem. Lett. (2005)

With A. Foroumadi, S. Emami, N. Rezvani & A. Asadipour. Synthesis of Certain Diarylsulfonylurea Derivatives As New Potential Antitumor Agents. Chem. Ind. J. 1(12):745-8, 2005

With L. Navidpour & R. Miri. Synthesis and calcium channel antagonist activity of new 1,4-dihydropyridine derivatives containing lipophilic 4-imidazolyl substituents. Arzneim. Forsch. (2004)

With O. Sabzevari, K. Abdi & M. Amini. Application of a simple and sensitive GC-MS method for determination of morphine in the hair of opium abusers. Anal. Bioanal. Chem. (2004)

With G. Amin & M. Iranshahi. A New Coumarin from Ferula persica. Pharmac. Biol. 42(6):440-3, 2004

With Y. Ghasemi, M. T. Yazdi, M. Amini, S. Shokravi & G. Zarrini. Parsiguine, A Novel Antimicrobial Substance from Fischerella ambigua. Pharmac. Biol. 42:318-22, 2004With V. Ziaee, H. Jalalizadeh & M. Iranshahi. Improved Synthesis of Vasicinone. Iran. J. Chem. & Chem. Eng. 23:33-36, 2004

With M. Amini & M. Khanavi. Simple High-Performance Liquid Chromatographic Method for Determination of Ciprofloxacin in Human Plasma. Iran. J. Pharm. Res. 2:99-101, 2004

With N. Rastkary & M. Sharifzadeh. Anticonvulsant Activities of New 1,4- Dihydropyridine Derivatives Containing 4-Nitroimidazolyl substituents. DARU 12:81-6, 2004

With S. Badakhshannoory & F. Hadizadeh. Assessment of Human AT1 Binding Affinity of some Novel 2-Alkylthio-1-[4-(N-a-Ethoxycarbonyl-Benzyl)Aminobenzyl]-5- Hydroxymethylimidazoles. DARU 12:31-5, 2004

With M.M. Akhavan, J.S. Mojarrad, A. Rouzrokh, S.A. Ebrahimi & M. Mahmoudian. Synthesis and antagonistic activity of four new 2-alkyl-N-biphenyl fused imidazoles on angiotensin II receptors. Farmaco (2003)

With A. Zarghi, A.H. Ebrahimabadi, F. Hassanzadeh & M.R. Heydari. Synthesis and anti-inflammatory activity of new 1-methyl-4-(4-X-benzenesulfonyl)pyrrolo[2,3-d] imidazole-5-carboxylates. Boll. Chim. Farmac. (2003)

With M. Iranshahi, G.R. Amin & H. Jalalizadeh. New Germacrane Derivative from Ferula perica. Pharmac. Biol. 41:431-3, 2003

With M. Amini & Hajmahmodi. Improved Chromatographic Method for Determination of Sodium Diclofenac in Injectable Solution and Prediction of Chemical Stability. J. Sci. Iran 14(1):21-5, 2003

With A. Zarghi, K. Derakhshandeh, F. Roshanzamir, M. Jorjani, H. Rastegar & M. Varmazyari. Synthesis and calcium antagonist activity of new 1,4-dihydropyridines containing nitrobenzylimidazolyl substituent in guinea-pig ileal smooth muscle. Boll. Chim. Farm. (2002)

With N. Rastkary, M. Jorjani & B. Shafaghi. Synthesis and Antihypertensive Activities of New 1, 4-Dihydropyridine Containing Nitroimidazolyl Substituent with a Nitrooxy Group at the 3-Ester Position. Archiv der Pharmazie (2002)

With A. Foroumadi, M. Mirzaei, S. Emami, P. Salari, F. Ghaffari & M. Amini. Synthesis and Antifungal Activity of Some New 1,2,4-Triazolo[3,4- b][1,3,4]thiadiazines. DARU 10:49-52, 2002

With M. Amini, A. Golabchifar, A.R. Dehpour & M.P. Hamedani. Synthesis and Calcium Channel Antagonist Activity of New 1,4-Dihydropyridine Derivatives Containing Dichloroimidazolyl Substituents. Arzneim Forsch Drug Res 52:21-26, 2002

With N. Rastkary, M. Jorjani & B. Shafaghi. Synthesis and Antihypertensive Activities of New 1,4-Dihydropyridine Containing Nitroimidazolyl Substituent with a Nitrooxy Group at the 3-Ester Position. Archiv der Pharmazie 2:69-79, 2002

With R. Miri, H. Niknahad, A. Vazin & A. Azarpira. Synthesis and Smooth Muscle Calcium Channel Antagonist Effects of New Derivatives of 1,4- Dihydropyridine Containing Nitroimidzolyl Substituent. DARU 10:130-6, 2002

With A. Foroumadi, M. Mirzaei, S. Emami, P. Salari, F. Ghaffari & M. Amini. Synthesis and Antifungal Activity of Some New 1,2,4-Triazolol[3,4- b][1,3,4]thiadiazines. DARU 10:34-7, 2001

With M. Abdollahi, M. Pirali, M. Karimi & M. Shahriarian. High performance liquid chromatography method for Determination of Nifedipine in Human Plasma. Daru 7(4): 1-4, 1999

With D. B. Bandarabadi, M.P. Hamedani & M. Amini. High Performance Liquid Chromatographic Method for Determination of Dipyridamole in Human Plasma. DARU 7 (1999)

With F. Hadizadeh, L. Karimi, M. Mahmoudian & N. Razzaghi. Synthesis and Angiotensin II Antagonist Activity of Novel 2-Arylthio-3-(2- alkyl-1-(4-carboxybenzyl)imidazolyl)acrylic acids. Pharm. Pharmacol. Commun 4, 1998

With G. Fanai. A Facile Synthesis of N-(4-Aryl-1,3-dithiol-2- ylidene)amides, and N-(4-Aryl-1,3-diselenol-2-ylidene)-amides. Synthesis (1984)

With G. Fanai. A Facile Synthesis of N-(4-Aryl-1,3-dithiol-2-ylidene)-amides, N-(4- or 5-Aryl-1,3,-thiaselenol-2-ylidene)-amides, and N-(4-Aryl-1,3,-diselenol-2-ylidene)- amides. Synthesis (1984)

With S. Sattari. Selenium Heterocycles XXXIII. Synthesis of Thieno[3,4-b]furan, Theino[3,4-b]indole and Seleno[3,4-b]indole, Four Novel Heterocycles. J. Heterocyclic Chem 19:227, 1982

With S. Sattari. A Facile Method for Acylation and Alkylation of Substituted Indoles. Synthesis (1981)

With G. Kiaeay. Chemistry of 1,2,3-Thiadiazole. IV. Synthesis of [1]Benzoxepino-[3,4-d][1,2,3]thiadiazole, [1]Benzothiepino-[3,4-d][1,2,3]thiadiazole, [1]Benzothiepino[4,3-d][1,2,3]thiadiazole, [1]Benzoxepino[4,3-d]oxadiazole, and [1]Benzoxepino[4,3-d]oxazole. Four Novel Heterocycles. J. Heterocyclic Chem 18:809, 1981

With G.Kiaeay & M. Vosooghi. Selenium Heterocycles XXXII. Synthesis of [1]Benzoxepino[3,4-d]-thiazole,[1]Benzothiepino[3,4-d]thiazole, [1]Benzoxepino[3,4-d]selenazole, and [1]Benzothiepino[3,4-d]selenazole. Four Novel Heterocycles. J. Heterocyclic Chem 18: 789, 1981

With A. Mazloumi & V. I. Cohen. Selenium Heterocycles XXVIII, Synthesis of pyrrolo[3,2-d]selenazole and Pyrrolo[3,2-d]thiazole. Two Novel Heterocycles. J. Heteroc. Chem 16:1563, 1979

With E. Behnam. Selenium Heterocycles XXVI. Synthesis of Thieno[3,4-b]benzofuran and Selenolo [3,4-b]benzofuran. Two Novel Heterocycles. J. Heteroc Chem, 15:589, 1978

With A. Mazloumi. Selenium Heterocycles XXVII. Synthesis of Thieno[3,4-d]thiazole and Selenolo[3,4-d]thiazole. Two Novel Heterocycles. J. Heterocyclic Chem 15:1455,1978

Selenium Heterocycles XXV. Synthesis of Thieno[3,4-b][1,2,3[thiadiazole, Selenolo[3,4-d][1,2,3]thiadiazole and Pyrrolo[3,4-d][1,2,3]thiadiazole. Three Novel Ring Systems. J. Heterocyclic Chem (1978)

With I. Lalezari & F. Savabi. A facile synthesis of 5-substituted 1,3 thiaselenole 2 thiones. Synthesis (1977)

With I. Lalezari & F. Savabi. A new synthesis of dimethyl-4-arylselenophene-2,3-dicarboxylates. Synthesis (1977)

Synthesis of 1,2,3-thiadiazolo [4,5-d]pyridazines. A new heterocyclic ring system. J. Heteroc. Chem. 13:301, 1976

With I. Lalezar & M. Yalpani. A simple New Synthesis of Arylalkynes Angew. Chem 9:46, 1970

A Novel Synthesis of Selenium Heterocycles: Substituted 1,2,3-selenadiazoles; Tetrahedron Lett (1969)